A novel, efficient synthesis of N-aryl pyrroles via reaction of 1-boronodienes with arylnitroso compounds.

نویسندگان

  • Fabien Tripoteau
  • Ludovic Eberlin
  • Mark A Fox
  • Bertrand Carboni
  • Andrew Whiting
چکیده

A one-pot hetero-Diels-Alder/ring contraction cascade is presented from the reaction of 1-boronodienes and arylnitroso derivatives to derive N-arylpyrroles in moderate to good yields (up to 82%).

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عنوان ژورنال:
  • Chemical communications

دوره 49 47  شماره 

صفحات  -

تاریخ انتشار 2013